Protocol

GLP-1 Titration Schedule

April 30, 2026
glp-1titrationsemaglutidetirzepatideretatrutideprotocol

Step-up reference for the three current GLP-1 family compounds. The package-insert cadence is the floor, not the target - for the dose-strategy framing (titrate-and-hold, when not to climb, what stops people on the cut), see the GLP-1 and Muscle Preservation article and Cycling Strategies.

Semaglutide (Wegovy / Ozempic / compounded)

Step Dose / week Hold
10.25 mg4 weeks
20.5 mg4 weeks
31.0 mg4 weeks
41.7 mg4 weeks
52.4 mgmaintenance (or hold lower if effective)

Slow-ramp variant: hold each step 6–8 weeks instead of 4 if GI tolerance is an issue. Skipping a step (e.g. 0.5 β†’ 1.7) routinely produces treatment-discontinuing nausea.

Tirzepatide (Zepbound / Mounjaro / compounded)

Step Dose / week Hold
12.5 mg4 weeks
25 mg4 weeks
37.5 mg4 weeks
410 mg4 weeks
512.5 mg4 weeks
615 mgmaintenance (or hold lower if effective)

Most operators stop climbing at 7.5 or 10 mg if fat loss is steady at 0.5–1% body weight per week. The 15 mg ceiling is for non-responders, not the default goal.

Retatrutide (investigational)

No approved label. Phase 2 (Jastreboff 2023) used once-weekly arms ranging from 1 mg to 12 mg with stepwise escalation. Community use mirrors the trial cadence:

Step Dose / week Hold
12 mg4 weeks
24 mg4 weeks
36 mg4 weeks
48 mg4 weeks
512 mgmaintenance ceiling (rarely needed)

Heart-rate elevation is the differentiator vs. GLP-1-only agents - track resting HR weekly. A sustained 8–10+ bpm increase warrants holding or dropping a step.

Split-dosing variant (all three)

  • Halve the weekly dose and inject twice weekly (e.g., 1.25 mg tirzepatide on Monday and Thursday instead of 2.5 mg once weekly).
  • Reduces peak serum concentration and the nausea that tracks with it. Keeps trough hunger from returning at end of week.
  • Off-label deviation from the half-life-driven schedule. Pharmacokinetically sound for these compounds because half-lives are 5–7 days; doesn’t work for shorter-half-life GLP-1s like liraglutide.

Climb / hold / drop rules

  • Climb only when fat loss has stalled (no scale or body-comp movement) for 2+ consecutive weeks at the current dose, AND side-effect tolerance is acceptable.
  • Hold indefinitely if the current dose is producing 0.5–1% body-weight loss per week. The lowest effective dose is the target, not the maximum.
  • Drop a step if nausea, vomiting or HR elevation is treatment-limiting. Climb back up only after a 4-week settle.
  • Maintenance taper after goal: drop to ~50% of the cutting dose for 6–12 months before considering discontinuation. Cold-stopping correlates with rebound; the maintenance phase is the protocol, not the afterthought.

Cross-references

GLP-1 Titration Schedule