Protocol

Melanotan II Loading Protocol

May 01, 2026
melanotan-iimt-iitanningprotocolloadingoperator-reference

Two-phase protocol: a 1–3 week loading ramp to saturate melanocytes while keeping nausea manageable, then weekly maintenance once the target shade is reached. For why MT-II works the way it does and where MC4R receptor desensitisation fits, see Melanocortin Map.

Pre-protocol checklist

  • Dermatology baseline. Photographic mole map at year zero is non-optional. MT-II darkens existing nevi and may precipitate new ones; a baseline is what makes the annual follow-up readable.
  • BAC water on hand. Reconstitution math in the Reconstitution Cheat Sheet; a 10 mg vial in 2 mL gives 50 mcg/u for clean unit math at 100/250/500 mcg doses.
  • Antihistamine. Cetirizine 10 mg or loratadine 10 mg 1 h before injection cuts the autonomic flush and a chunk of the nausea.
  • UV plan. 20–30 min UV exposure 2–3x/week is required for the protocol to produce a tan. MT-II raises melanin capacity; UV oxidises it.

Loading phase

DayDoseNotes
1–3100 mcg / day SCTest response. Inject pre-bed to sleep through the nausea peak.
4–6250 mcg / day SCAntihistamine 1 h before. UV starting from week 1 if tolerated.
7+500 mcg / day SCContinue daily until target shade is reached, typically 1–3 weeks.

Operators who tolerate poorly hold each step for 4–6 days instead of 3. Skipping a step (e.g. 100 → 500 mcg) reliably produces severe nausea, vomiting, and flushing strong enough that some users stop the protocol entirely.

Maintenance phase

PatternDoseWhy
Weekly 500 mcg – 1 mg once per week Once saturation is reached, pigment persists months. Weekly dosing keeps the signal alive without re-triggering load-phase nausea.
Bi-weekly 500 mcg every 2 weeks For users who reach saturation easily; cuts cost and dose load further. Watch the shade and bump back to weekly if it fades.

UV pairing rules

  • Without UV the protocol fails. MT-II without sun or a tanning bed produces grey-tinged or no visible tan. The melanin is there; UV is the activator.
  • Start UV from week 1. Building tolerance to dose and UV in parallel is faster than loading first and adding UV later.
  • 20–30 minute sessions, 2–3x/week. Standard moderate-exposure tanning cadence. Don’t double up - MT-II enhances melanin response, not UV protection.
  • SPF still applies. Sun damage isn’t turned off by enhanced pigmentation. SPF 30+ on face and any non-target areas.

Side-effect management

  • Nausea / flush: antihistamine 1 h before; inject pre-bed; eat something small with carbs 30 min before injection.
  • Spontaneous erections: common at first injections, fades with continued use. Time injection so the next 4–6 hours are private.
  • Dark moles: expected. New small moles are common. Discuss anything unusual with the dermatologist on the annual follow-up.
  • Decreased appetite: mild, often welcome on a cut. Not the goal of the protocol but a frequent side-effect.

What stops people

  • Skipping the loading ramp. 500 mcg cold first dose produces vomiting and treatment-discontinuing nausea. The ramp is short; respect it.
  • Skipping UV. The most common reason MT-II “doesn’t work” in user reports. Without UV, the pigment doesn’t express on the skin in a useful way.
  • Stacking with PDE5 inhibitors at high doses. Synergistic erection effect; priapism risk if both are dosed close together at high doses. See Stacking Safety Quick Reference.
  • Skipping the dermatology baseline. A year of MT-II use without a pre-protocol mole map makes the annual follow-up much harder to read. Five minutes once is worth it.

Cross-references

Melanotan II Loading Protocol